SCHEMBL7329993

SCHEMBL7329993

N=C(N)c1ccc(NCc2ccccc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 2/20 0.74
PRSS1 P07477 10/20 0.59
F2 P00734 5/20 0.59
F10 P00742 3/20 0.59
F7 P08709 3/20 0.59
CA1 P00915 2/20 0.57
CA2 P00918 2/20 0.57
PRSS2 P07478 2/20 0.56
PRSS3 P35030 2/20 0.56
TMPRSS6 Q8IU80 2/20 0.56
ST14 Q9Y5Y6 2/20 0.56
KLK1 P06870 2/20 0.55
KLK5 Q9Y337 2/20 0.55
HTT P42858 1/20 0.55
F12 P00748 1/20 0.52
F3 P13726 1/20 0.52
PKM P14618 1/20 0.52
CA12 O43570 1/20 0.51
CA9 Q16790 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14259897 0.88 PRSS1 (0.59) MRGPRX1PRSS1F2F10F7
SCHEMBL1924100 0.80 HTT (0.78) CA1CA2HTTCA12CA9
SCHEMBL2742815 0.78 CA1 (0.70) CA1CA2HTTCA12CA9
SCHEMBL1446643 0.78 CA1 (0.70) CA1CA2HTTCA12CA9
SCHEMBL14259895 0.78 PRSS1 (0.53) MRGPRX1PRSS1F2F10F7
SCHEMBL28778912 0.77 CA1 (0.64) CA1CA2HTTCA12CA9
N-Benzylaniline SCHEMBL28146501 0.77 FFAR1 (0.62) CA1CA2HTTCA12CA9
SCHEMBL3875680 0.77 PRSS1 (0.84) PRSS1F2F10PRSS2PRSS3
SCHEMBL12348324 0.77 PRSS1 (0.70) PRSS1F2F10PRSS2PRSS3
SCHEMBL11882481 0.76 CA1 (0.58) MRGPRX1CA1CA2HTTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5550159-A Peptide mimics useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1996-08-27 US disclosed
US-5453440-A Amidine functional group on benzene ring, anticoagulants G. D. SEARLE & CO. (US) 1995-09-26 US disclosed
WO-1993018058-A1 PEPTIDES MIMICS USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-09-16 WO disclosed