SCHEMBL733229

SCHEMBL733229

C=CCC(C)(C)COC(=O)N[C@H](C(=O)N1C[C@H](Oc2nccc3cc(OC)c(C=C)cc23)C[C@H]1C(=O)OCC)C1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
ELANE P08246 1/20 0.37
KCNH2 Q12809 1/20 0.37
CTSB P07858 2/20 0.34
PPP3CB P16298 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3624949 0.94 CYP3A4 (0.40) CYP3A4ELANEKCNH2CTSBPPP3CB
SCHEMBL731547 0.94 CYP3A4 (0.39) CYP3A4ELANEKCNH2CTSBPPP3CB
SCHEMBL10081455 0.91 CYP3A4 (0.37) CYP3A4ELANEKCNH2CTSB
SCHEMBL1243486 0.89 CYP3A4 (0.37) CYP3A4ELANEKCNH2CTSB
SCHEMBL1244279 0.88 CYP3A4 (0.37) CYP3A4ELANEKCNH2CTSBPPP3CB
SCHEMBL3618649 0.87 CYP3A4 (0.40) CYP3A4ELANEKCNH2CTSBPPP3CB
SCHEMBL8195028 0.84 CYP3A4 (0.36) CYP3A4ELANEKCNH2PDE4APDE4B
SCHEMBL733230 0.83 CYP3A4 (0.33) CYP3A4ELANEKCNH2
SCHEMBL14562633 0.82 CYP3A4 (0.38) CYP3A4ELANEKCNH2CTSBPPP3CB
SCHEMBL14562561 0.81 CYP3A4 (0.38) CYP3A4ELANEKCNH2CTSBPPP3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079479-B1 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2014-11-26 EP disclosed
US-8138164-B2 HCV NS3 protease inhibitors MERCK SHARP & DOHME CORP. (US) 2012-03-20 US disclosed