SCHEMBL7339557

SCHEMBL7339557

OCc1cnc2sccn12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.49
CHEK1 O14757 1/20 0.49
LIMK1 P53667 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
KDM4E B2RXH2 9/20 0.47
HSD17B10 Q99714 9/20 0.44
ALDH1A1 P00352 8/20 0.44
HPGD P15428 7/20 0.44
RECQL P46063 1/20 0.44
MAPT P10636 6/20 0.42
MAPK1 P28482 1/20 0.42
TDP1 Q9NUW8 1/20 0.39
TSHR P16473 4/20 0.39
PKM P14618 1/20 0.39
NPC1 O15118 5/20 0.38
RAB9A P51151 5/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
TP53 P04637 1/20 0.38
HTT P42858 1/20 0.36
KMT2A Q03164 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2628994 0.69
SCHEMBL15401844 0.69
SCHEMBL5045177 0.69
SCHEMBL7328706 0.69 IDO1 (0.44) DYRK1A
SCHEMBL269609 0.69 CHEK1 (0.62) DYRK1ACHEK1LIMK1CLK4KDM4E
SCHEMBL14976996 0.68 CHEK1 (0.51) DYRK1ACHEK1LIMK1CLK4KDM4E
SCHEMBL13066867 0.67 KDM4E (0.43) DYRK1ACHEK1LIMK1CLK4KDM4E
SCHEMBL766237 0.66 CHEK1 (1.00) DYRK1ACHEK1LIMK1CLK4KDM4E
SCHEMBL7494643 0.65 DYRK1A (0.39) DYRK1ACHEK1LIMK1CLK4KDM4E
SCHEMBL9609565 0.65 KDM4E (0.47) DYRK1ACHEK1LIMK1CLK4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191124-B1 VIRICIDES PHARMACIA & UPJOHN COMPANY 2001-02-20 US disclosed
EP-0757692-A1 METHANOL DERIVATIVES FOR TREATMENT OF RETROVIRAL INFECTIONS ESPECIALLY HIV INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-12 EP disclosed
WO-1995029922-A1 METHANOL DERIVATIVES FOR TREATMENT OF RETROVIRAL INFECTIONS ESPECIALLY HIV INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-09 WO disclosed
EP-0463212-A1 Imidazo[2,1-b]thiazole compound anti-ulcer agent containing the same NIKKEN CHEMICALS CO., LTD. (JP) 1992-01-02 EP disclosed