SCHEMBL7344217

SCHEMBL7344217

O=C(NCCN1CCCCC1)[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(=O)[C@H](Cc1ccc(Br)cc1)NC(=O)N1CCCCCC1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 8/20 0.52
ITGB3 P05106 1/20 0.49
ITGA2B P08514 1/20 0.49
HRH3 Q9Y5N1 3/20 0.49
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CACNA1B Q00975 2/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
NPY1R P25929 1/20 0.46
EGFR P00533 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343687 0.93 TACR2 (0.53) TACR2ITGB3ITGA2BHRH3NPC1
SCHEMBL7337619 0.91 CACNA1B (0.57) TACR2CACNA1B
SCHEMBL7340969 0.91 CACNA1B (0.57) TACR2CACNA1B
SCHEMBL7336892 0.90 TACR2 (0.54) TACR2ITGB3ITGA2BHRH3NPC1
SCHEMBL7346404 0.89 TACR2 (0.50) TACR2ITGB3ITGA2BNPC1RAB9A
SCHEMBL7349125 0.89 TACR2 (0.50) TACR2ITGB3ITGA2BCACNA1B
SCHEMBL7340850 0.88 TACR2 (0.49) TACR2ITGB3ITGA2BCACNA1BEGFR
SCHEMBL7341412 0.86 TACR2 (0.58) TACR2ITGB3ITGA2BCACNA1B
SCHEMBL7345251 0.86 TACR2 (0.60) TACR2CACNA1B
SCHEMBL7342593 0.86 TACR2 (0.58) TACR2CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed