SCHEMBL7345954

SCHEMBL7345954

CC(C)C[C@H](NC(=O)N1CCCCCC1)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NCCCN1CCN(C)CC1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 12/20 0.56
CACNA1B Q00975 6/20 0.54
ITGB3 P05106 1/20 0.52
ITGA2B P08514 1/20 0.52
CTSS P25774 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7341412 0.96 TACR2 (0.58) TACR2CACNA1BITGB3ITGA2BCTSS
SCHEMBL7337619 0.91 CACNA1B (0.57) TACR2CACNA1BCTSS
SCHEMBL7340969 0.91 CACNA1B (0.57) TACR2CACNA1BCTSS
SCHEMBL7340635 0.91 CACNA1B (0.56) TACR2CACNA1BCTSS
SCHEMBL7341622 0.89 PLG (0.58) TACR2CACNA1BCTSS
SCHEMBL7343417 0.89 CACNA1B (0.58) CACNA1BCTSS
SCHEMBL7341276 0.89 CACNA1B (0.58) CACNA1BCTSS
SCHEMBL7345251 0.88 TACR2 (0.60) TACR2CACNA1BCTSS
SCHEMBL7337268 0.87 TACR2 (0.61) TACR2ITGB3ITGA2B
SCHEMBL7345374 0.87 CACNA1B (0.66) CACNA1BITGB3ITGA2BCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0546389-B1 Piperidylmethyl substituted chroman derivatives as agents for the treatment of diseases of the central nervous system BAYER AG (DE) 1996-04-17 EP disclosed
EP-0546388-B1 Azaheterocyclylmethyl-chromans as agents for the treatment of diseases of the central nervous system BAYER AG (DE) 1996-03-27 EP disclosed
EP-0546389-A1 Piperidylmethyl substituted chroman derivatives as agents for the treatment of diseases of the central nervous system BAYER AG (DE) 1993-06-16 EP disclosed
EP-0546388-A1 Azaheterocyclylmethyl-chromans as agents for the treatment of diseases of the central nervous system BAYER AG (DE) 1993-06-16 EP disclosed