SCHEMBL7346196

SCHEMBL7346196

CC(C(=O)O)C1Cc2ccc(O)cc2NC1=O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.41
LMNA P02545 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.35
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
MAPT P10636 1/20 0.34
BLM P54132 1/20 0.34
CYP2D6 P10635 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
MAPK1 P28482 1/20 0.34
OPRK1 P41145 2/20 0.33
OPRM1 P35372 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28114452 0.76 ESR2 (0.46) ESR2LMNAALDH1A1CYP3A4BRD4
SCHEMBL4621828 0.72 ESR2 (0.43) ESR2LMNAALDH1A1CYP3A4TSHR
SCHEMBL7212449 0.71 ESR2 (0.42) ESR2LMNAALDH1A1CYP3A4TSHR
SCHEMBL7073390 0.71 GAA (0.42) ESR2LMNAALDH1A1CYP3A4TSHR
SCHEMBL17049180 0.70 ESR2 (0.39) ESR2LMNAALDH1A1CYP3A4TSHR
SCHEMBL27725432 0.70 ESR2 (0.73) ESR2LMNAALDH1A1BRD4CREBBP
SCHEMBL3412848 0.69 NQO2 (0.44) ESR2LMNATSHRCYP2D6
SCHEMBL17049187 0.68 KDM4E (0.50) ESR2LMNAALDH1A1TSHRMAPT
SCHEMBL17413603 0.68 GAA (0.64) ESR2MAPTOPRK1
SCHEMBL17055844 0.68 ESR2 (0.36) ESR2LMNAALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971878-A1 AMINE COMPOUNDS, THEIR PRODUCTION AND USE AS AMYLOID-BETA PRODUCTION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2000-01-19 EP disclosed
WO-1998038156-A1 AMINE COMPOUNDS, THEIR PRODUCTION AND USE AS AMYLOID-BETA PRODUCTION INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-03 WO disclosed