SCHEMBL7350586

SCHEMBL7350586

Nc1nccc(N2CCC(N3C(=O)OC4C(C5CCC(C(=O)O)CC5)CCCC43)CC2)n1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.41
HRH4 Q9H3N8 1/20 0.35
PDE4D Q08499 1/20 0.35
BTK Q06187 1/20 0.34
NEK2 P51955 2/20 0.33
KDM4E B2RXH2 1/20 0.31
CYP2C19 P33261 1/20 0.31
CCNC P24863 1/20 0.31
CDK8 P49336 1/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL7350589 0.91 HRH3 (0.42) HRH3HRH4PDE4DBTKCCNC
SCHEMBL7344255 0.88 HRH3 (0.42) HRH3HRH4PDE4DBTKNEK2
SCHEMBL27513356 0.84 HRH3 (0.39) HRH3HRH4PDE4DBTKNEK2
SCHEMBL27496064 0.78 HRH3 (0.40) HRH3HRH4PDE4DBTK
SCHEMBL7344262 0.78 HRH3 (0.40) HRH3HRH4PDE4D
SCHEMBL7341730 0.73 KDM4E (0.35) KDM4ECYP2C19
SCHEMBL7342860 0.73 ALK (0.42)
SCHEMBL7350171 0.73 HRH4 (0.45) HRH4KDM4E
SCHEMBL8356693 0.72 HRH3 (0.40) HRH3HRH4PDE4DBTKNEK2
SCHEMBL7367195 0.72 PARP1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1219933-A Novel oxazolidine derivatives, process for their preparation and pharmaceutical preparations containing these compounds BOEHRINGER MANNHEIM GMBH (DE) 1999-06-16 CN disclosed
EP-0891359-A1 NOVEL OXAZOLIDINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION AND MEDICAMENTS CONTAINING THEM Roche Diagnostics GmbH (DE) 1999-01-20 EP disclosed
WO-1997036899-A1 NOVEL OXAZOLIDINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION AND MEDICAMENTS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1997-10-09 WO disclosed