SCHEMBL7352242

SCHEMBL7352242

CCCCCCN(Cc1ccc2ccccc2c1)c1c(N[C@@H](Cc2ccccc2)C(=O)OC)c(=O)c1=O

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.45
ITGA4 P13612 5/20 0.45
HDAC1 Q13547 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
PPARG P37231 2/20 0.40
PPARD Q03181 2/20 0.40
PPARA Q07869 2/20 0.40
BCHE P06276 1/20 0.39
BIRC2 Q13490 1/20 0.39
F2 P00734 1/20 0.39
CNR2 P34972 1/20 0.38
POLB P06746 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352253 1.00 ITGB1 (0.45) ITGB1ITGA4HDAC1HDAC6PPARG
SCHEMBL7357178 0.92 ITGB1 (0.51) ITGB1ITGA4BCHE
SCHEMBL7357187 0.92 ITGB1 (0.51) ITGB1ITGA4BCHE
SCHEMBL7361891 0.88 ITGB1 (0.51) ITGB1ITGA4BIRC2CNR2POLB
SCHEMBL7361897 0.88 ITGB1 (0.51) ITGB1ITGA4BIRC2CNR2POLB
SCHEMBL7348616 0.87 ITGB1 (0.46) ITGB1ITGA4BIRC2CNR2POLB
SCHEMBL7348625 0.87 ITGB1 (0.46) ITGB1ITGA4BIRC2CNR2POLB
SCHEMBL7353260 0.82 ITGB1 (0.54) ITGB1ITGA4
SCHEMBL7362260 0.80 ITGB1 (0.57) ITGB1ITGA4
SCHEMBL7362255 0.80 ITGB1 (0.57) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166050-A 3,4-diamino-3-cyclobutene-1,2-dione derivatives which inhibit leukocyte adhesion mediated by VLA-4 AMERICAN HOME PRODUCTS CORPORATION (US) 2000-12-26 US disclosed