SCHEMBL7353572

SCHEMBL7353572

CCC(NC(=NC#N)Nc1ccc(N)nc1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 2/20 0.38
HDAC3 O15379 5/20 0.37
HDAC1 Q13547 5/20 0.37
HDAC8 Q9BY41 3/20 0.37
TACR3 P29371 6/20 0.37
TACR2 P21452 1/20 0.37
HDAC4 P56524 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC2 Q92769 2/20 0.35
NCOR2 Q9Y618 2/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ROCK2 O75116 2/20 0.34
ROCK1 Q13464 2/20 0.34
TRPV1 Q8NER1 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7354758 1.00 QPCT (0.38) QPCTHDAC3HDAC1HDAC8TACR3
SCHEMBL7353557 1.00 QPCT (0.38) QPCTHDAC3HDAC1HDAC8TACR3
SCHEMBL7353564 1.00 QPCT (0.38) QPCTHDAC3HDAC1HDAC8TACR3
SCHEMBL8622425 0.88 QPCT (0.39) QPCTHDAC3HDAC1HDAC8TACR3
SCHEMBL7424824 0.88 QPCT (0.39) QPCTHDAC3HDAC1HDAC8TACR3
SCHEMBL8620009 0.88 QPCT (0.39) QPCTHDAC3HDAC1HDAC8TACR3
SCHEMBL7349710 0.85 QPCT (0.37) QPCTHDAC3HDAC1HDAC8TACR3
SCHEMBL7349700 0.85 QPCT (0.37) QPCTHDAC3HDAC1HDAC8TACR3
SCHEMBL7349695 0.85 QPCT (0.37) QPCTHDAC3HDAC1HDAC8TACR3
SCHEMBL7356810 0.82 KMT2A (0.47) TACR3KDM4ELMNAROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655057-B1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS UPJOHN CO (US) 1997-09-17 EP claimed
US-5567722-A DIURETICS THE UPJOHN COMPANY (US) 1996-10-22 US claimed
WO-1994004500-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS THE UPJOHN COMPANY (US) 1994-03-03 WO claimed
EP-0655057-B1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS UPJOHN CO (US) 1997-09-17 EP disclosed
US-5567722-A DIURETICS THE UPJOHN COMPANY (US) 1996-10-22 US disclosed
WO-1994004500-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS THE UPJOHN COMPANY (US) 1994-03-03 WO disclosed