SCHEMBL7355245

SCHEMBL7355245

CCN(C)C1CCCN(C(=O)c2ccc(NC(=O)c3ccccc3C)cc2)c2ccc(C)cc21

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 7/20 0.70
AVPR2 P30518 6/20 0.70
AVPR1B P47901 2/20 0.70
ABCB11 O95342 1/20 0.70
HTR1A P08908 1/20 0.70
CHRM1 P11229 1/20 0.70
OXTR P30559 1/20 0.70
SLC6A4 P31645 1/20 0.70
ADRA1A P35348 1/20 0.70
OPRM1 P35372 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7345848 0.91 AVPR1A (0.83) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL7383625 0.83 AVPR2 (0.63) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL7352677 0.83 AVPR1A (0.80) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL7348782 0.83 AVPR1A (0.80) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL7353668 0.83 AVPR1A (0.80) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL7348322 0.83 AVPR1A (0.77) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL7353531 0.83 AVPR1A (0.64) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL7352805 0.82 AVPR1A (0.79) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL7353026 0.82 AVPR1A (0.79) AVPR1AAVPR2AVPR1BABCB11HTR1A
SCHEMBL7346631 0.82 AVPR1A (0.79) AVPR1AAVPR2AVPR1BABCB11HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846514-A Enhancement of the efficacy of nifedipine by deuteration ISOTECHNIKA, INC. (CA) 1998-12-08 US disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed