SCHEMBL7355895

SCHEMBL7355895

O=C(O)[C@@H]1CCN2C(=O)CC[C@H](NC(=O)[C@H](Br)Cc3ccccc3)C(=O)N2C1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACE P12821 16/20 0.55
MME P08473 14/20 0.55
ACE2 Q9BYF1 3/20 0.41
MMP2 P08253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7355833 0.85 ACE (0.52) ACEMMEACE2MMP2
SCHEMBL7347578 0.85 ACE (0.52) ACEMMEACE2MMP2
SCHEMBL7348441 0.84 ACE (0.54) ACEMME
SCHEMBL8317625 0.80 ACE (0.79) ACEMME
SCHEMBL9312905 0.80 ACE (0.79) ACEMME
SCHEMBL7352272 0.79 MME (0.45) ACEMME
SCHEMBL7380923 0.71 ACE (1.00) ACEMMEACE2
SCHEMBL7345704 0.71 ACE (1.00) ACEMMEACE2
SCHEMBL7351462 0.71 ACE (0.78) ACEMME
SCHEMBL7374154 0.71 ACE (0.78) ACEMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640086-A1 NOVEL MERCAPTOACETYLAMIDO PYRIDAZO 1,2]PYRIDAZINE, PYRAZOLO 1,2]PYRIDAZINE, PYRIDAZO 1,2-a] 1,2]DIAZEPINE AND PYRAZOLO 1,2-a] 1,2]DIAZEPINE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE MERRELL PHARMACEUTICALS INC. (US) 1995-03-01 EP disclosed
WO-1993023403-A1 NOVEL MERCAPTOACETYLAMIDO PYRIDAZO[1,2]PYRIDAZINE, PYRAZOLO[1,2]PYRIDAZINE, PYRIDAZO[1,2-a][1,2]DIAZEPINE AND PYRAZOLO[1,2-a][1,2]DIAZEPINE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE MERRELL DOW PHARMACEUTICALS INC. (US) 1993-11-25 WO disclosed