SCHEMBL7358756

SCHEMBL7358756

CCCCCc1c(N(C)C)ccc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 3/20 0.51
KDM4E B2RXH2 6/20 0.42
MAPT P10636 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
TLR8 Q9NR97 4/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
ALDH1A1 P00352 5/20 0.40
GAA P10253 5/20 0.40
NPC1 O15118 4/20 0.40
HTT P42858 4/20 0.40
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
GLA P06280 1/20 0.40
RCE1 Q9Y256 1/20 0.40
CNR1 P21554 2/20 0.39
CNR2 P34972 1/20 0.39
HPGD P15428 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2125551 0.81 CYP1A2 (0.48) NCEH1KDM4EMAPTTDP1TLR8
SCHEMBL6919402 0.79 NCEH1 (0.47) NCEH1KDM4EMAPTTDP1TLR8
SCHEMBL8671922 0.79 CYP1A2 (0.47) NCEH1KDM4EMAPTTLR8MEN1
SCHEMBL2127033 0.79 CYP1A2 (0.47) NCEH1KDM4EMAPTTLR8MEN1
SCHEMBL2125169 0.79 CYP1A2 (0.47) NCEH1KDM4EMAPTTLR8MEN1
SCHEMBL11381159 0.78 TYR (0.47) NCEH1KDM4EMAPTTDP1TLR8
SCHEMBL10800999 0.78 NCEH1 (0.46) NCEH1KDM4EMAPTTDP1TLR8
SCHEMBL284699 0.78 TYR (0.47) NCEH1KDM4EMAPTTDP1TLR8
SCHEMBL2126531 0.78 NCEH1 (0.49) NCEH1KDM4EMAPTTLR8ALDH1A1
SCHEMBL283786 0.78 TYR (0.47) NCEH1KDM4EMAPTTDP1TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4556676-A Antidepressant derivatives of trans-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine PFIZER INC. (US) 1985-12-03 US disclosed
US-4536518-A Antidepressant derivatives of cis-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine PFIZER INC. (US) 1985-08-20 US disclosed
EP-0030081-B1 ANTIDEPRESSANT DERIVATIVES OF CIS-4-PHENYL-1,2,3,4-TETRAHYDRO-1-NAPHTHALENAMINE AND PHARMACEUTICAL COMPOSITIONS THEREOF PFIZER INC. (US) 1983-03-02 EP disclosed
EP-0028901-A1 Antidepressant derivatives of trans-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine and pharmaceutical compositions thereof PFIZER INC. (US) 1981-05-20 EP disclosed