SCHEMBL7359166

SCHEMBL7359166

COc1ccc(CCN(C)CCC(=O)Nc2cc(OC)c(OC)c(OC)c2)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.68
KMT2A Q03164 4/20 0.66
MEN1 O00255 2/20 0.66
GAA P10253 2/20 0.66
ALDH1A1 P00352 1/20 0.66
MAPT P10636 1/20 0.66
HPGD P15428 1/20 0.66
CYP1A2 P05177 1/20 0.59
CYP2D6 P10635 1/20 0.59
BLM P54132 1/20 0.58
PMP22 Q01453 1/20 0.58
LMNA P02545 5/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
NPC1 O15118 2/20 0.50
KDM4E B2RXH2 1/20 0.50
RAB9A P51151 1/20 0.49
BMP1 P13497 1/20 0.48
BCHE P06276 1/20 0.48
ACHE P22303 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7326215 0.85 CYP3A4 (0.67) CYP3A4KMT2AMEN1GAAALDH1A1
SCHEMBL7335360 0.84 CYP3A4 (0.62) CYP3A4KMT2AMEN1GAAALDH1A1
SCHEMBL7360114 0.84 CYP3A4 (0.64) CYP3A4KMT2AMEN1GAAALDH1A1
SCHEMBL7323568 0.82 CYP3A4 (0.64) CYP3A4KMT2AMEN1GAAALDH1A1
SCHEMBL10338948 0.81 CYP3A4 (0.74) CYP3A4KMT2AMEN1GAAALDH1A1
SCHEMBL9491941 0.81 CYP3A4 (0.61) CYP3A4KMT2AMEN1GAAALDH1A1
SCHEMBL7359187 0.80 KMT2A (0.58) KMT2AMEN1ALDH1A1MAPTLMNA
SCHEMBL7175914 0.79 CYP3A4 (0.74) CYP3A4KMT2AMEN1GAAALDH1A1
SCHEMBL7355951 0.78 CYP3A4 (0.54) CYP3A4KMT2AMEN1GAAALDH1A1
SCHEMBL9195021 0.78 SCN1A (0.54) KMT2AMEN1GAAALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0852142-A1 Diamines in the treatment of arrhythmia SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1998-07-08 EP disclosed
EP-0639973-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1995-03-01 EP disclosed
WO-1993023024-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1993-11-25 WO disclosed