SCHEMBL7359864

SCHEMBL7359864

NC(=O)C[C@H](NC(=O)CC1CCCC1)C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.43
KMT2A Q03164 2/20 0.43
EPHX1 P07099 2/20 0.43
ECE1 P42892 1/20 0.41
AAK1 Q2M2I8 1/20 0.38
NPC1 O15118 4/20 0.37
RAB9A P51151 3/20 0.37
EPHX2 P34913 2/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
ERCC1 P07992 1/20 0.35
ERCC4 Q92889 1/20 0.35
CTSD P07339 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359870 1.00 HPGD (0.43) HPGDKMT2AEPHX1ECE1AAK1
SCHEMBL5274437 0.87 KMT2A (0.45) HPGDKMT2AEPHX1ECE1AAK1
SCHEMBL5274432 0.87 KMT2A (0.45) HPGDKMT2AEPHX1ECE1AAK1
SCHEMBL4134832 0.81 CNR2 (0.43) HPGDKMT2AEPHX1SMN1; SMN2CTSD
SCHEMBL4145751 0.80 PSEN1 (0.44) HPGDKMT2AEPHX1AAK1EPHX2
SCHEMBL5275391 0.75 EPHX2 (0.44) HPGDKMT2AEPHX1NPC1RAB9A
SCHEMBL5275396 0.75 EPHX2 (0.44) HPGDKMT2AEPHX1NPC1RAB9A
SCHEMBL7882899 0.72 KMT2A (0.53) HPGDKMT2AEPHX1NPC1RAB9A
SCHEMBL10808220 0.72 HPGD (0.42) HPGDKMT2AEPHX1AAK1NPC1
SCHEMBL24158323 0.72 HPGD (0.47) HPGDKMT2ANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1268117-A Novel inhibitors of aggrecanase and matrix metalloproteinases for the treatment of arthritis DU PONT PHARM CO (US) 2000-09-27 CN claimed
EP-1005448-A2 NOVEL INHIBITORS OF AGGRECANASE AND MATRIX METALLOPROTEINASES FOR THE TREATMENT OF ARTHRITIS Du Pont Pharmaceuticals Company (US) 2000-06-07 EP disclosed
WO-1999009000-A2 NOVEL INHIBITORS OF AGGRECANASE AND MATRIX METALLOPROTEINASES FOR THE TREATMENT OF ARTHRITIS DU PONT PHARMACEUTICALS COMPANY (US) 1999-02-25 WO disclosed