SCHEMBL7362685

SCHEMBL7362685

CN(C)c1ccc(C(=O)c2cnn3c(-c4ccncc4)ccnc23)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 2/20 0.49
MAP2K1 Q02750 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
DYRK1B Q9Y463 1/20 0.49
TLR8 Q9NR97 1/20 0.44
FYN P06241 1/20 0.44
MAPT P10636 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
PIM1 P11309 4/20 0.43
LIMK1 P53667 2/20 0.43
GSK3A P49840 3/20 0.42
MAPK13 O15264 2/20 0.42
MARK2 Q7KZI7 2/20 0.42
EPHA2 P29317 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366385 0.88 MAP2K1 (0.49) ALDH1A1KDM4EMAP2K1CLK4DYRK1B
SCHEMBL7361917 0.85 KDM4E (0.69) ALDH1A1KDM4EMAP2K1CLK4DYRK1B
SCHEMBL5790981 0.84 CLK4 (0.64) ALDH1A1KDM4EMAP2K1CLK4DYRK1B
SCHEMBL7402736 0.81 KDM4E (0.67) KDM4ETLR8BRAF
SCHEMBL7367609 0.80 MAP2K1 (0.55) ALDH1A1KDM4EMAP2K1CLK4DYRK1B
SCHEMBL7362641 0.80 TLR8 (0.52) ALDH1A1KDM4EMAP2K1CLK4DYRK1B
SCHEMBL10941570 0.79 CLK4 (0.55) ALDH1A1KDM4EMAP2K1CLK4DYRK1B
SCHEMBL7362738 0.78 CLK4 (0.73) ALDH1A1KDM4EMAP2K1CLK4DYRK1B
SCHEMBL7366580 0.78 MAP2K1 (0.55) ALDH1A1KDM4EMAP2K1CLK4DYRK1B
SCHEMBL1879312 0.77 TLR8 (0.49) ALDH1A1KDM4EMAP2K1CLK4DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed