SCHEMBL7364645

SCHEMBL7364645

CC(C)CCN(C)[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)N1CCC(O)CC1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 11/20 0.55
YAP1 P46937 5/20 0.45
CTSK P43235 1/20 0.45
UTS2R Q9UKP6 1/20 0.44
MME P08473 1/20 0.43
ACE P12821 1/20 0.43
CPA1 P15085 1/20 0.43
ACE2 Q9BYF1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195243 0.91 CACNA1B (0.59) CACNA1BYAP1MMEACECPA1
SCHEMBL7399075 0.91 CACNA1B (0.51) CACNA1BMMEACECPA1ACE2
SCHEMBL7398580 0.90 CACNA1B (0.50) CACNA1BYAP1CTSKMMEACE
SCHEMBL7402922 0.89 CACNA1B (0.49) CACNA1BUTS2RMMEACECPA1
SCHEMBL7343479 0.84 CACNA1B (0.55) CACNA1BYAP1MMEACECPA1
SCHEMBL7402336 0.83 CACNA1B (0.55) CACNA1BYAP1
SCHEMBL8188856 0.82 UTS2R (0.54) YAP1UTS2R
SCHEMBL5833508 0.82 CACNA1B (0.52) CACNA1BYAP1MMEACECPA1
SCHEMBL7408660 0.82 UTS2R (0.59) UTS2R
SCHEMBL7405382 0.82 CACNA1B (0.57) CACNA1BYAP1MMEACECPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO claimed
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed