SCHEMBL7366032

SCHEMBL7366032

Cc1ccc(-c2n[nH]c(=O)c3ncccc23)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 5/20 0.49
ALDH1A1 P00352 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ATM Q13315 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
COMT P21964 1/20 0.46
PDE9A O76083 1/20 0.44
HPGD P15428 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAP2K4 P45985 4/20 0.43
MAPKAPK3 Q16644 3/20 0.43
MAPK6 Q16659 3/20 0.43
MAPKAPK2 P49137 2/20 0.43
MAPKAPK5 Q8IW41 2/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369415 0.90 ATM (0.49) MAPK1ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL3652876 0.86 NPSR1 (0.64) ALDH1A1MEN1KMT2ASMN1; SMN2ATM
SCHEMBL2886126 0.84 GSK3A (0.52) MAPK1ALDH1A1MEN1KMT2AHPGD
SCHEMBL7362195 0.81 MAP2K4 (0.57) MAPK1ALDH1A1ATMNPSR1HPGD
SCHEMBL7362532 0.80 MAP2K4 (0.53) MAPK1ATMNPSR1MAP2K4MAPKAPK3
SCHEMBL7368649 0.80 MAPK1 (0.70) MAPK1ALDH1A1SMN1; SMN2HPGDMAP2K4
SCHEMBL1786578 0.79 ATM (0.73) MAPK1ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL19153217 0.79 PARP1 (0.49) CYP1A2L3MBTL1PARP1TSHRNPC1
SCHEMBL16535289 0.78 LRRK2 (0.61) ALDH1A1SMN1; SMN2ATMNPSR1HPGD
SCHEMBL17887975 0.76 ITK (0.59) MAPK1ALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed