SCHEMBL7366104

SCHEMBL7366104

CCOc1noc(CO)c1C

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
CHRM3 P20309 3/20 0.35
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
S1PR1 P21453 3/20 0.33
S1PR3 Q99500 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26926708 0.79 HTR2A (0.36) HTR2AHTR2CCHRM3CHRM2CHRM4
SCHEMBL10157747 0.78
SCHEMBL7374475 0.75 HTR2A (0.41) HTR2AHTR2CCHRM3CHRM2CHRM4
SCHEMBL12385469 0.70
SCHEMBL7160156 0.69 CA12 (0.38) HTR2AHTR2CCHRM3CHRM2CHRM4
SCHEMBL7165046 0.68 HTR2A (0.36) HTR2AHTR2CCHRM3CHRM2CHRM4
SCHEMBL7374814 0.65 TP53 (0.43)
SCHEMBL26926744 0.64 HTR2A (0.36) HTR2AHTR2CCHRM3CHRM2CHRM4
SCHEMBL10157729 0.64 PTGS1 (0.31)
SCHEMBL4933992 0.64 HTR2A (0.39) HTR2AHTR2CCHRM3CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994107-A1 5-Arylisoxazol-4-yl-substituted 2-amino carboxylic acid compounds H. LUNDBECK A/S (DK) 2000-04-19 EP disclosed
EP-0726896-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1996-08-21 EP disclosed
WO-1995012587-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1995-05-11 WO disclosed