SCHEMBL7366555

SCHEMBL7366555

CC(=O)Nc1cccc(-c2cccc(-n3c(=O)c(Cc4cccnc4O)nc4cccnc43)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.42
AKT1 P31749 7/20 0.42
AKT2 P31751 6/20 0.42
AKT3 Q9Y243 6/20 0.42
CYP2C9 P11712 3/20 0.42
TP53 P04637 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
STAT1 P42224 1/20 0.40
CYP17A1 P05093 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
RXFP1 Q9HBX9 2/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
MCHR1 Q99705 1/20 0.38
MEN1 O00255 1/20 0.38
MAPK10 P53779 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6801778 0.85 EGFR (0.45) TGFBR1AKT1AKT2AKT3CYP2C9
SCHEMBL7366554 0.83 EGFR (0.41) TGFBR1AKT1AKT2AKT3CYP2C9
SCHEMBL6797247 0.82 EGFR (0.53) AKT1AKT2AKT3CYP2C9TP53
SCHEMBL6797690 0.82 EGFR (0.46) AKT1AKT2AKT3TP53CYP17A1
SCHEMBL6798795 0.80 EGFR (0.49) AKT1AKT2AKT3CYP2C9TP53
SCHEMBL6800418 0.80 AKT1 (0.43) AKT1AKT2AKT3TP53NPC1
Hydrochloric Acid SCHEMBL6796872 0.78 EGFR (0.43) AKT1AKT2AKT3CYP2C9TP53
SCHEMBL6799820 0.78 TP53 (0.47) AKT1TP53RXFP1MCHR1MEN1
SCHEMBL6801892 0.78 EGFR (0.44) AKT1TP53NPC1SMN1; SMN2EGFR
SCHEMBL6804831 0.77 NPC1 (0.44) TP53NPC1RAB9ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874845-A1 PYRIDO (2,3-B) PYRAZINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-11-04 EP disclosed
WO-1997024355-A1 PYRIDO (2,3-B) PYRAZINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-07-10 WO disclosed