SCHEMBL7366612

SCHEMBL7366612

O=C(C=Cc1ccc([N+](=O)[O-])cc1)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.82

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.82
PTPN12 Q05209 1/20 0.82
PTPN22 Q9Y2R2 1/20 0.82
MAOB P27338 7/20 0.76
BCHE P06276 1/20 0.76
MAPT P10636 6/20 0.70
HSPD1 P10809 1/20 0.68
HSPE1 P61604 1/20 0.68
ALDH1A1 P00352 5/20 0.67
LMNA P02545 4/20 0.67
CYP1B1 Q16678 1/20 0.67
HTT P42858 2/20 0.65
NTSR1 P30989 1/20 0.64
MAOA P21397 4/20 0.63
RAB9A P51151 1/20 0.62
TGM2 P21980 1/20 0.61
CYP19A1 P11511 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7454702 1.00 PTPN1 (0.82) PTPN1PTPN12PTPN22MAOBBCHE
SCHEMBL9779522 0.91 MAPT (0.84) PTPN1PTPN12PTPN22MAOBBCHE
SCHEMBL9779526 0.91 MAPT (0.84) PTPN1PTPN12PTPN22MAOBBCHE
SCHEMBL9338320 0.90 PTPN1 (0.76) PTPN1PTPN12PTPN22MAOBBCHE
SCHEMBL30301794 0.90 PTPN1 (0.76) PTPN1PTPN12PTPN22MAOBBCHE
SCHEMBL31441210 0.90 MAPT (0.86) PTPN1PTPN12PTPN22MAOBBCHE
SCHEMBL1073090 0.90 MAPT (0.86) PTPN1PTPN12PTPN22MAOBBCHE
SCHEMBL1073092 0.90 MAPT (0.86) PTPN1PTPN12PTPN22MAOBBCHE
SCHEMBL31441212 0.90 MAPT (0.86) PTPN1PTPN12PTPN22MAOBBCHE
SCHEMBL32681391 0.89 MAOB (0.72) PTPN1PTPN12PTPN22MAOBBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892780-B1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-11-20 EP disclosed
US-5942544-A α-branched anilines, toluenes, and analogs thereof as factor Xa inhibitors DUPONT PHARMACEUTICALS COMPANY (US) 1999-08-24 US disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed
US-3989708-A HYPOTENSIVE, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-11-02 US disclosed