Cerdulatinib

Cerdulatinib

SCHEMBL736734

CCS(=O)(=O)N1CCN(c2ccc(Nc3ncc(C(N)=O)c(NC4CC4)n3)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

JAK1JAK3SYKTYK2

The experimentally established mechanism targets of Cerdulatinib. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK known ✓ P43405 20/20 1.00
JAK1 known ✓ P23458 3/20 1.00
TYK2 known ✓ P29597 2/20 1.00
JAK3 known ✓ P52333 2/20 1.00
CHEK1 O14757 2/20 1.00
RET P07949 2/20 1.00
FLT3 P36888 2/20 1.00
RPS6KA3 P51812 2/20 1.00
MAPK10 P53779 2/20 1.00
STK4 Q13043 2/20 1.00
STK3 Q13188 2/20 1.00
MARK2 Q7KZI7 2/20 1.00
TBK1 Q9UHD2 2/20 1.00
RPS6KA6 Q9UK32 2/20 1.00
JAK2 O60674 2/20 1.00
NUAK1 O60285 1/20 1.00
CSF1R P07333 1/20 1.00
FLT4 P35916 1/20 1.00
MAP3K9 P80192 1/20 1.00
ITK Q08881 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cerdulatinib SCHEMBL29462019 0.99 SYK (1.00) SYKJAK1CHEK1RETTYK2
SCHEMBL737349 0.92 SYK (1.00) SYKJAK1CHEK1RETTYK2
SCHEMBL8737323 0.92 SYK (0.85) SYKJAK1CHEK1RETTYK2
SCHEMBL20734854 0.92 SYK (0.85) SYKJAK1CHEK1RETTYK2
SCHEMBL21554052 0.91 SYK (0.83) SYKJAK1CHEK1RETTYK2
SCHEMBL736830 0.91 SYK (1.00) SYKJAK1CHEK1RETTYK2
SCHEMBL21554059 0.91 SYK (0.82) SYKJAK1CHEK1RETTYK2
SCHEMBL21554086 0.90 SYK (0.82) SYKJAK1CHEK1RETTYK2
SCHEMBL17076550 0.89 SYK (0.81) SYKJAK1CHEK1RETTYK2
SCHEMBL22030443 0.89 SYK (0.81) SYKJAK1CHEK1RETTYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2292 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137953-A1 METHOD FOR TARGETED TREATING DERMATOSES STRATA SKIN SCIENCES INC. (US) 2026-05-21 US claimed
WO-2026090557-A1 SYSTEMS AND METHODS FOR PROCESSING ISM AND MCAS CLINICAL TRIAL DATA TELIOS PHARMA INC. (US) 2026-04-30 WO claimed
US-12611408-B2 Methods for treating nail brittleness, fragility, or pitting CHEMISTRY RX (US) 2026-04-28 US claimed
US-20260097056-A1 SYK ACTIVATORS AND INHIBITORS IN NEURODEGENERATIVE DISEASES UNIV VIRGINIA PATENT FOUNDATION (US) 2026-04-09 US claimed
US-20260097028-A1 Methods of Treating Myeloproliferative Neoplasms KARTOS THERAPEUTICS INC (US) 2026-04-09 US claimed
US-20260008791-A1 CHEMICAL COMPOUNDS BORAH INC (US) 2026-01-08 US claimed
US-20260008856-A1 METHODS OF TREATING DISEASE USING ANTI-IL1RAP ANTIBODIES AND ANTIBODY DRUG CONJUGATES BLUEFIN BIOMEDICINE INC (US) 2026-01-08 US claimed
US-20250382312-A1 BORON CONTAINING PYRAZOLE COMPOUNDS, COMPOSITIONS COMPRISING THEM, METHODS AND USES THEREOF BORAH INC (US) 2025-12-18 US claimed
US-20250367113-A1 DRUG DELIVERY SYSTEM COMPRISING AN ANTI-INFLAMMATORY AGENT OR A SALT THEREOF FOR THE APPLICATION TO ESOPHAGEAL MUCOUS MEMBRANES ESOCAP AG (CH) 2025-12-04 US claimed
EP-4640714-A2 METHODS FOR ASSESSING RISK OF DEVELOPING A VIRAL DISEASE USING A GENETIC TEST PML Screening, LLC (US) 2025-10-29 EP claimed
EP-3942045-A1 A DBAIT MOLECULE IN COMBINATION WITH KINASE INHIBITOR FOR THE TREATMENT OF CANCER ONXEO (FR) 2022-01-26 EP claimed
WO-2019113475-A1 TOPICAL OINTMENT FORMULATIONS AND THEIR USE IN TREATING SKIN CONDITIONS Dermavant Sciences GmbH (CH) 2019-06-13 WO claimed
WO-2018189566-A1 USE OF A CHEMICAL COMPOUND AS A THERAPEUTIC AGENT BEVEC DORIAN (DE) 2018-10-18 WO claimed
EP-3191098-A1 COMBINATIONS AND DOSING REGIMES TO TREAT RB-POSITIVE TUMORS G1 Therapeutics, Inc. (US) 2017-07-19 EP claimed
EP-2321283-B1 2,6-DIAMINO-PYRIMIDIN-5-YL-CARBOXAMIDES AS SYK OR JAK KINASES INHIBITORS PORTOLA PHARM INC (US) 2016-07-13 EP claimed
WO-2016040858-A1 COMBINATIONS AND DOSING REGIMES TO TREAT RB-POSITIVE TUMORS G1 THERAPEUTICS, INC. (US) 2016-03-17 WO claimed
CN-102066340-B 2, 6-diamino-pyrimidin- 5-yl-carboxamides as SRK or JAK kinases inhibitors PORTOLA PHARM INC 2014-05-14 CN claimed
US-20130237493-A1 COMBINATION THERAPY OF 4-(CYCLOPROPYLAMINO)-2-(4-(4-(ETHYLSULFONYL)PIPERAZIN-1-YL)PHENYLAMINO)PYRIMIDINE-5-CARBOXAMIDE AND FLUDARABINE PORTOLA PHARMACEUTICALS, INC. (US) 2013-09-12 US claimed
EP-2621489-A1 COMBINATIONS OF 4-(CYCLOPROPYLAMINO)-2-(4-(4-(ETHYLSULFONYL)PIPERAZIN-1-YL)PHENYLAMINO)PYRIMIDINE-5-CARBOXAMIDE AND FLUDARABINE Portola Pharmaceuticals, Inc. (US) 2013-08-07 EP claimed
WO-2012045020-A1 COMBINATIONS OF 4-(CYCLOPROPYLAMINO)-2-(4-(4-(ETHYLSULFONYL)PIPERAZIN-1-YL)PHENYLAMINO)PYRIMIDINE-5-CARBOXAMIDE AND FLUDARABINE PORTOLA PHARMACEUTICALS, INC. (US) 2012-04-05 WO claimed