SCHEMBL7367344

SCHEMBL7367344

CC(C)(O)c1cc(Cl)c(CNC(=O)c2cccnc2Oc2cncc(Cl)c2)s1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 5/20 0.48
POLB P06746 1/20 0.42
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7406034 0.92 MAPK8 (0.51) MAPK8GAA
SCHEMBL7372538 0.88 MAPK8 (0.53) MAPK8GAA
SCHEMBL7369180 0.83 MAPK8 (0.47) MAPK8
SCHEMBL7373396 0.82 MAPK8 (0.55) MAPK8
SCHEMBL7368839 0.81 MAPK8 (0.48) MAPK8POLBGAA
SCHEMBL7371907 0.80 MAPK8 (0.48) MAPK8POLBGAA
SCHEMBL7370770 0.80 MAPK8 (0.50) MAPK8POLB
SCHEMBL7370304 0.79 HPGD (0.62) MAPK8POLBGAA
SCHEMBL7369860 0.78 MAPK8 (0.50) MAPK8POLB
SCHEMBL7373226 0.77 MAPK8 (0.49) MAPK8POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380218-B1 FOR THERAPY OF RESPIRATORY, ALLERGIC, AND INFLAMMATORY DISORDERS COMPRISING ASTHMA, CHRONIC OBSTRUCTIVE PULMONARY DISEASE, ACUTE RESPIRATORY DISEASE SYNDROME, PULMONARY HYPERSENSITIVITY, AND ALLERGIC RHINITIS IN A MAMMAL PFIZER INC 2002-04-30 US disclosed
EP-0971894-A1 NICOTINAMIDE DERIVATIVES Pfizer Products Inc. (US) 2000-01-19 EP disclosed
WO-1998045268-A1 NICOTINAMIDE DERIVATIVES PFIZER PRODUCTS INC. (US) 1998-10-15 WO disclosed