SCHEMBL7368620

SCHEMBL7368620

COc1cc(C(=O)c2ccc(Cl)cc2)cc([N+](=O)[O-])c1O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 5/20 0.64
MAPT P10636 4/20 0.55
HPGD P15428 2/20 0.55
LMNA P02545 2/20 0.55
ALDH1A1 P00352 1/20 0.55
RAF1 P04049 1/20 0.55
MAPK1 P28482 1/20 0.55
GFER P55789 1/20 0.55
PAX8 Q06710 1/20 0.55
ABCC3 O15438 1/20 0.54
ABCC4 O15439 1/20 0.54
NR1I2 O75469 1/20 0.54
ABCB11 O95342 1/20 0.54
NR3C1 P04150 1/20 0.54
PGR P06401 1/20 0.54
HTR1A P08908 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
RARB P10826 1/20 0.54
COMT P21964 1/20 0.54
SLC6A2 P23975 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7373740 0.88 TTR (0.71) TTRMAPTHPGDLMNAALDH1A1
SCHEMBL7371341 0.88 TTR (0.65) TTRMAPTHPGDLMNAALDH1A1
SCHEMBL7365333 0.87 TTR (0.75) TTRMAPTHPGDLMNAALDH1A1
SCHEMBL7369400 0.86 TTR (0.67) TTRMAPTHPGDLMNAALDH1A1
SCHEMBL7365244 0.86 TTR (0.60) TTRMAPTHPGDLMNAALDH1A1
SCHEMBL7203416 0.85 HPGD (0.59) TTRMAPTHPGDLMNAALDH1A1
SCHEMBL31443266 0.84 CNR1 (0.67) MAPTHPGDLMNAALDH1A1MAPK1
SCHEMBL7369924 0.84 TTR (0.64) TTRMAPTHPGDLMNAALDH1A1
SCHEMBL7371244 0.84 TTR (0.71) TTRMAPTHPGDLMNAALDH1A1
SCHEMBL8466506 0.82 TTR (0.78) TTRMAPTHPGDLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5476875-A Catechol derivatives HOFFMAN-LA ROCHE INC. (US) 1995-12-19 US disclosed
US-5236952-A Inhibit the enzyme catechol-O-methyltransferase; for treatment of Parkinson's disease administered with L-dopa HOFFMANN-LA ROCHE INC. (US) 1993-08-17 US disclosed
EP-0237929-B1 3,5-DISUBSTITUTED PYROCATECHOL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-06-02 EP disclosed
EP-0237929-A1 3,5-Disubstituted pyrocatechol derivatives F. HOFFMANN-LA ROCHE AG (CH) 1987-09-23 EP disclosed