SCHEMBL7374656

SCHEMBL7374656

Cc1ccc(-c2ccccc2C(=O)Nc2ccc(C(=O)N(C)c3ccccc3OCCCCCN3CCN(C)CC3)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
AVPR2 P30518 10/20 0.48
AVPR1A P37288 3/20 0.47
AVPR1B P47901 2/20 0.47
EGFR P00533 1/20 0.43
KDR P35968 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374907 1.00 KDM4E (0.49) KDM4EALDH1A1POLBAVPR2AVPR1A
SCHEMBL7377133 1.00 KDM4E (0.49) KDM4EALDH1A1POLBAVPR2AVPR1A
Hydrochloric Acid SCHEMBL7749380 0.99 KDM4E (0.48) KDM4EALDH1A1POLBAVPR2AVPR1A
SCHEMBL7376990 0.99 KDM4E (0.49) KDM4EALDH1A1POLBAVPR2AVPR1A
Hydrochloric Acid SCHEMBL7376857 0.98 KDM4E (0.49) KDM4EALDH1A1POLBAVPR2AVPR1A
SCHEMBL7377877 0.97 AVPR2 (0.49) KDM4EALDH1A1POLBAVPR2AVPR1A
SCHEMBL7372942 0.90 AVPR2 (0.46) AVPR2AVPR1AAVPR1B
SCHEMBL7751053 0.90 AVPR2 (0.46) AVPR2AVPR1AAVPR1B
SCHEMBL7372097 0.89 AVPR2 (0.46) AVPR2AVPR1AAVPR1B
SCHEMBL7375946 0.89 NPSR1 (0.42) ALDH1A1AVPR2AVPR1AAVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed