SCHEMBL7375809

SCHEMBL7375809

CC(C)(C)OC(=O)CC[C@@](NC(=O)[C@@H](CSC(=O)c1ccccc1)Cc1ccccc1)(Nc1ccccc1)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 5/20 0.40
CYP3A4 P08684 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ABCC3 O15438 1/20 0.40
NR1I2 O75469 1/20 0.40
ABCB11 O95342 1/20 0.40
NR3C1 P04150 1/20 0.40
RARG P13631 1/20 0.40
CNR1 P21554 1/20 0.40
OPRK1 P41145 1/20 0.40
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
NR1I3 Q14994 1/20 0.40
CTSS P25774 2/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7291272 0.88 CYP1A2 (0.38) PPARACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7284671 0.88 CYP1A2 (0.38) PPARACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7370508 0.86 CYP1A2 (0.37) PPARACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7290272 0.85 MME (0.43) ACE
SCHEMBL7283576 0.82 CYP1A2 (0.39) PPARACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7283663 0.82 CYP3A4 (0.35) PPARACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7283657 0.82 CYP3A4 (0.35) PPARACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL9400825 0.82 CYP3A4 (0.35) PPARACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7378978 0.80 CYP3A4 (0.34) PPARACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7283659 0.80 ECE1 (0.38) PPARACYP3A4CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0341081-B1 Novel amino acid derivatives ONO PHARMACEUTICAL CO (JP) 1995-07-05 EP disclosed
US-5317021-A Analgesics, anticonvulsants ONO PHARMACEUTICAL CO., LTD. (JP) 1994-05-31 US disclosed
US-5202340-A Analgesics, anticonvulsants, anxiolytic agents, inhibitors for enkephalinases ONO PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
US-5017589-A Analgesic, antianxiety, anticonvulsant ONO PHARMACEUTICAL CO., LTD. (JP) 1991-05-21 US disclosed