SCHEMBL7377205

SCHEMBL7377205

CCOC(=O)CCNCCc1ccc(Cl)cc1CN1CCC[C@H]1C(=O)NC(=O)[C@](C)(O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
RECQL P46063 1/20 0.44
F2 P00734 7/20 0.44
F10 P00742 3/20 0.38
GPBAR1 Q8TDU6 3/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CNR2 P34972 2/20 0.35
PPARD Q03181 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CNR1 P21554 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7372915 0.84 F2 (0.56) F2F10GPBAR1CNR2CNR1
SCHEMBL7379417 0.84 F2 (0.48) TSHRMAPK1RECQLF2GPBAR1
SCHEMBL7373230 0.83 F2 (0.47) TSHRMAPK1RECQLF2GPBAR1
SCHEMBL7374615 0.82 F2 (0.62) F2F10
SCHEMBL7377776 0.81 F2 (0.48) TSHRMAPK1RECQLF2F10
SCHEMBL6921255 0.81 F2 (0.69) F2F10ALDH1A1
SCHEMBL7380524 0.79 F2 (0.53) TSHRMAPK1RECQLF2F10
SCHEMBL7378295 0.74 F2 (0.62) F2F10GPBAR1
SCHEMBL7452387 0.73 F2 (0.52) F2F10GPBAR1ALDH1A1
SCHEMBL6921253 0.72 F2 (0.36) F2F10SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002050056-A1 BENZYLAMINE DERIVATIVES AND THEIR USE AS THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-06-27 WO disclosed