SCHEMBL7377396

SCHEMBL7377396

O=C(O)C1CCCCN1C(=O)CCS

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACE P12821 6/20 0.62
LMNA P02545 2/20 0.50
HSD17B10 Q99714 2/20 0.50
CYP2C19 P33261 1/20 0.50
KDM4E B2RXH2 1/20 0.50
F2 P00734 1/20 0.50
REN P00797 1/20 0.50
LTA4H P09960 1/20 0.50
MAPT P10636 1/20 0.50
PEPD P12955 1/20 0.50
ALOX15 P16050 1/20 0.50
PTGS1 P23219 1/20 0.50
HTR2A P28223 1/20 0.50
PTGS2 P35354 1/20 0.50
HRH1 P35367 1/20 0.50
THPO P40225 1/20 0.50
PMP22 Q01453 1/20 0.50
ACE2 Q9BYF1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6789982 0.95 ACE (0.69) ACELMNAHSD17B10CYP2C19KDM4E
SCHEMBL683432 0.95 ACE (0.69) ACELMNAHSD17B10CYP2C19KDM4E
SCHEMBL6789984 0.95 ACE (0.69) ACELMNAHSD17B10CYP2C19KDM4E
SCHEMBL7381767 0.90 ACE (0.55) ACELMNAHSD17B10CYP2C19KDM4E
SCHEMBL7377569 0.87 ACE (0.54) ACELMNAHSD17B10CYP2C19KDM4E
SCHEMBL7381081 0.86 ACE (0.56) ACELMNAHSD17B10CYP2C19KDM4E
SCHEMBL3048970 0.85 ACE (0.60) ACELMNAHSD17B10CYP2C19KDM4E
SCHEMBL6782701 0.83 ACE (0.72) ACEREN
SCHEMBL6782705 0.83 ACE (0.72) ACEREN
SCHEMBL12249655 0.81 ACE (0.56) ACEREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0012845-B1 TETRAHYDROISOQUINOLINE COMPOUNDS, PROCESS FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Tanabe Seiyaku Co., Ltd. (JP) 1983-06-22 EP disclosed
US-4154840-A Antihypertensive pipecolic acid derivatives E. R. SQUIBB & SONS, INC. (US) 1979-05-15 US disclosed
US-4105776-A ANGIOTENSIN CONVERTING ENZYME INHIBITORS, HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1978-08-08 US disclosed
US-4046889-A HYPOTENSIVE AGENTS, ENZYME INHIBITORS, ANGIOTENSIN CONVERSION E. R. SQUIBB & SONS, INC. (US) 1977-09-06 US disclosed