SCHEMBL7384141

SCHEMBL7384141

CC(C)CC(C(=O)O)N(CCc1cncn1Cc1ccccc1[N+](=O)[O-])C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.37
CYP2C19 P33261 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7375020 0.86 CYP11B1 (0.39) CYP11B1CYP11B2
SCHEMBL3715232 0.86 CYP11B1 (0.39) CYP11B1CYP11B2
SCHEMBL7374943 0.85 CYP11B1 (0.39) ALDH1A1KDM4ELMNACYP2C19CYP11B1
SCHEMBL7382224 0.85 CYP11B1 (0.41) LMNACYP11B1CYP11B2
SCHEMBL7379194 0.84 ACE2 (0.42) CYP11B1CYP11B2
SCHEMBL7398066 0.84 CYP11B1 (0.37) ALDH1A1KDM4ETDP1CYP11B1CYP11B2
SCHEMBL7384484 0.82 CYP11B1 (0.41) ALDH1A1KDM4ELMNATDP1POLB
SCHEMBL7383285 0.82 ACE2 (0.38) CYP11B1CYP11B2
SCHEMBL3686724 0.82 CYP11B1 (0.35) CYP11B1CYP11B2
SCHEMBL1655292 0.81 CYP11B1 (0.36) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed
EP-1183019-A2 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF Millennium Pharmaceuticals, Inc. (US) 2002-03-06 EP disclosed
WO-2000066104-A2 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2000-11-09 WO disclosed