SCHEMBL7384144

SCHEMBL7384144

CC(C)CC(NCC(C(=O)O)c1cncn1Cc1ccccc1[N+](=O)[O-])C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
POLB P06746 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
ACE2 Q9BYF1 4/20 0.38
ACE P12821 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7375023 0.85 ACE2 (0.39) POLBACE2ACE
SCHEMBL3715236 0.85 ACE2 (0.39) KDM4EACE2ACESMN1; SMN2
SCHEMBL7382228 0.85 ACE2 (0.43) POLBMAPTACE2ACE
SCHEMBL7374947 0.85 ACE2 (0.39) ALDH1A1CYP2C19MAPTACE2ACE
SCHEMBL7379198 0.83 ACE2 (0.46) ALDH1A1KDM4EMAPTHTTACE2
SCHEMBL7398069 0.83 P2RY14 (0.38) ALDH1A1KDM4ETDP1CYP2C19ACE2
SCHEMBL7375034 0.83 ANPEP (0.43) ALDH1A1KDM4ETDP1ACE2ACE
SCHEMBL7384489 0.82 ACE2 (0.43) ALDH1A1KDM4ETDP1CYP2C19MAPT
SCHEMBL3707154 0.81 CD274 (0.42) ACE2ACE
SCHEMBL7383288 0.81 ACE2 (0.41) ACE2ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed
EP-1183019-A2 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF Millennium Pharmaceuticals, Inc. (US) 2002-03-06 EP disclosed
WO-2000066104-A2 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2000-11-09 WO disclosed