SCHEMBL7396137

SCHEMBL7396137

COc1ccc(S(=O)(=O)n2cnc3c2c(=O)n(CC2CC2)c(=O)n3CC2CC2)cc1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 19/20 0.69
PDE4B Q07343 19/20 0.69
PDE4C Q08493 19/20 0.69
PDE4D Q08499 19/20 0.69
PDE5A O76074 17/20 0.69
ADORA3 P0DMS8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400203 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7399392 0.82 PDE4A (0.79) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7397039 0.79 PDE5A (0.66) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL8058416 0.77 PDE4A (0.70) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7400585 0.74 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7451032 0.72 PDE5A (1.00) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7390028 0.72 PDE4A (0.92) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7392224 0.72 PDE4A (0.61) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9350631 0.70 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7436549 0.70 PDE5A (0.79) PDE4APDE4BPDE4CPDE4DPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563168-B1 XANTHINE DERIVATIVES BEECHAM GROUP PLC (GB) 2000-07-05 EP claimed
EP-0563168-B1 XANTHINE DERIVATIVES BEECHAM GROUP PLC (GB) 2000-07-05 EP disclosed
US-5409934-A Antiallergens BEECHAM GROUP P.L.C. (GB) 1995-04-25 US disclosed
EP-0563168-A1 XANTHINE DERIVATIVES BEECHAM GROUP PLC (GB) 1993-10-06 EP disclosed
WO-1992011260-A1 XANTHINE DERIVATIVES BEECHAM GROUP PLC (GB) 1992-07-09 WO disclosed