SCHEMBL7396409

SCHEMBL7396409

Cc1ccncc1-c1cccc(F)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.57
GRM5 P41594 1/20 0.49
CYP17A1 P05093 6/20 0.49
CYP1A2 P05177 4/20 0.49
CYP11B1 P15538 3/20 0.49
CYP11B2 P19099 3/20 0.49
TDO2 P48775 1/20 0.49
RPS6KA3 P51812 1/20 0.48
ABL1 P00519 1/20 0.47
PTGES2 Q9H7Z7 1/20 0.45
CYP3A4 P08684 1/20 0.45
CDC7 O00311 1/20 0.44
ROCK2 O75116 1/20 0.44
MAP4K4 O95819 1/20 0.44
PIM1 P11309 1/20 0.44
PRKACA P17612 1/20 0.44
CDK2 P24941 1/20 0.44
GSK3B P49841 1/20 0.44
HIPK2 Q9H2X6 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2421428 0.82 RPS6KA3 (0.57) CYP17A1CYP1A2CYP11B1CYP11B2RPS6KA3
SCHEMBL6744647 0.80 RPS6KA3 (0.63) SLC22A12CYP17A1CYP11B1CYP11B2RPS6KA3
SCHEMBL26462958 0.79 ABL1 (0.50) CYP17A1CYP1A2CYP11B1CYP11B2RPS6KA3
SCHEMBL11627241 0.79 MEN1 (0.56) CYP17A1CYP1A2CYP11B1CYP11B2ABL1
SCHEMBL30494154 0.79 ABL1 (0.50) CYP17A1CYP1A2CYP11B1CYP11B2RPS6KA3
SCHEMBL7396406 0.79 SLC22A12 (0.54) SLC22A12CYP17A1CYP11B1CYP11B2RPS6KA3
SCHEMBL30494314 0.79 ABL1 (0.50) CYP17A1CYP1A2CYP11B1CYP11B2RPS6KA3
SCHEMBL26103090 0.79 CYP11B1 (0.46) CYP17A1CYP1A2CYP11B1CYP11B2RPS6KA3
SCHEMBL30494189 0.79 CYP11B1 (0.46) CYP17A1CYP1A2CYP11B1CYP11B2RPS6KA3
SCHEMBL27876161 0.79 PDE4B (0.56) SLC22A12CYP17A1CYP1A2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1123933-A1 2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]chromane as CNS active agent MERCK PATENT GmbH (DE) 2001-08-16 EP disclosed
EP-0707007-A1 Amino(thio)ether derivatives as CNS active agents MERCK PATENT GmbH (DE) 1996-04-17 EP disclosed