SCHEMBL7397165

SCHEMBL7397165

CC[C@H](C)[C@H](NC(=O)[C@H](CC(=O)O)NC(C)=O)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(=O)O)C(N)=O)[C@@H](C)CC

nearest known ligand 0.73

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 1/20 0.73
MAGI3 Q5TCQ9 1/20 0.60
CCKBR P32239 13/20 0.58
CCKAR P32238 2/20 0.58
CASP1 P29466 1/20 0.54
CASP3 P42574 1/20 0.54
CASP4 P49662 1/20 0.54
CASP5 P51878 1/20 0.54
CASP7 P55210 1/20 0.54
CASP9 P55211 1/20 0.54
CASP6 P55212 1/20 0.54
CASP8 Q14790 1/20 0.54
CASP10 Q92851 1/20 0.54
MMP2 P08253 2/20 0.53
ECE1 P42892 1/20 0.53
MMP9 P14780 1/20 0.53
MMP8 P22894 1/20 0.53
MMP1 P03956 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9069917 0.97 EDNRA (0.69) EDNRAMAGI3CCKBRCCKARCASP1
SCHEMBL7396826 0.95 EDNRA (0.69) EDNRAMAGI3CCKBRCCKARCASP1
SCHEMBL7396823 0.95 EDNRA (0.69) EDNRAMAGI3CCKBRCCKARCASP1
SCHEMBL7400880 0.95 EDNRA (0.69) EDNRAMAGI3CCKBRCCKARCASP1
SCHEMBL30533185 0.93 EDNRA (0.82) EDNRAMAGI3CASP1CASP3CASP4
SCHEMBL7395342 0.92 EDNRA (0.81) EDNRAMAGI3ECE1
SCHEMBL7395344 0.92 EDNRA (0.81) EDNRAMAGI3ECE1
SCHEMBL7401708 0.91 EDNRA (0.61) EDNRAMAGI3CCKBRCCKARCASP1
SCHEMBL7397607 0.91 EDNRA (0.72) EDNRAMAGI3CCKBRCCKARCASP1
SCHEMBL9069770 0.91 MAGI3 (0.68) EDNRAMAGI3CCKBRCCKARCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5504070-A ADMINISTERING OLIGOPEPTIDES, PHOSPHONATES AND MODIFIED AMINO ACIDS AS INHIBITORS BERLEX LABORATORIES, INC. (US) 1996-04-02 US claimed
US-5504070-A ADMINISTERING OLIGOPEPTIDES, PHOSPHONATES AND MODIFIED AMINO ACIDS AS INHIBITORS BERLEX LABORATORIES, INC. (US) 1996-04-02 US disclosed
WO-1993011154-A1 INHIBITORS OF THE CONVERSION OF BIG ENDOTHELIN TO ENDOTHELIN BERLEX LABORATORIES, INC. (US) 1993-06-10 WO disclosed