SCHEMBL7399788

SCHEMBL7399788

COc1ccccc1/C=C/c1nc2c([nH]1)c(=O)n(C)c(=O)n2C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.53
LCK P06239 1/20 0.53
LYN P07948 1/20 0.53
SRC P12931 1/20 0.53
CSK P41240 1/20 0.53
BTK Q06187 1/20 0.53
PTK6 Q13882 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399791 1.00 ABL1 (0.53) ABL1LCKLYNSRCCSK
SCHEMBL7315144 0.90
SCHEMBL7401304 0.90
SCHEMBL7304364 0.85 KDM4E (0.63)
SCHEMBL7311852 0.84
SCHEMBL7304947 0.84
SCHEMBL7315091 0.82
SCHEMBL7301067 0.82
SCHEMBL7302584 0.81
SCHEMBL7304617 0.81 KDM4E (0.52) ABL1LCKLYNSRCCSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861405-A A2-SELECTIVE ADENOSINE RECEPTOR ANTAGONIST AS ANTIDEPRESSANTS AND CNS STIMULANTS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1999-01-19 US disclosed
WO-1994025462-A1 8-SUBSTITUTED 1,3,7-TRIALKYL-XANTHINE DERIVATIVES AS A2-SELECTIVE ADENOSINE RECEPTOR ANTAGONISTS THE UNITED STATES OF AMERICA, REPRESENTED BY THE (US) 1994-11-10 WO disclosed