SCHEMBL7400221

SCHEMBL7400221

N#Cc1c(OCCC2CCCCN2)nc(N)nc1-c1ccco1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.46
ADORA1 P30542 8/20 0.46
ADORA2B P29275 5/20 0.46
CCNA2 P20248 2/20 0.43
CDK2 P24941 2/20 0.43
CCNA1 P78396 2/20 0.43
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 3/20 0.38
GAA P10253 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ADORA3 P0DMS8 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
SMARCA2 P51531 1/20 0.36
ERAP1 Q9NZ08 1/20 0.36
USP2 O75604 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445430 0.78 ADORA1 (0.50) ADORA2AADORA1ADORA2BCCNA2CDK2
SCHEMBL6441743 0.77 ADORA1 (0.56) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL6440638 0.77 ADORA2A (0.56) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL5046621 0.76 ADORA2A (0.55) ADORA2AADORA1ADORA2BCCNA2CDK2
SCHEMBL5046844 0.75 ADORA1 (0.60) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL5037058 0.75 ADORA2A (0.60) ADORA2AADORA1ADORA2BCCNA2CDK2
SCHEMBL6449356 0.75 ADORA2A (0.54) ADORA2AADORA1ADORA2BCCNA2CDK2
SCHEMBL6441656 0.75 ADORA1 (0.49) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL5036930 0.74 ADORA2A (0.59) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL6441085 0.73 ADORA2A (0.58) ADORA2AADORA1ADORA2BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1261327-A2 ADENOSINE RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2002-12-04 EP disclosed
WO-2001062233-A2 ADENOSINE RECEPTOR MODULATORS F. HOFFMANN LA ROCHE AG (CH) 2001-08-30 WO disclosed