SCHEMBL7400569

SCHEMBL7400569

Cc1cc(NC(=O)c2ccccc2-c2cccnc2)ccc1C(=O)N1Cc2cccnc2Oc2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 7/20 0.48
ROCK2 O75116 1/20 0.44
TP53 P04637 1/20 0.44
SHMT2 P34897 1/20 0.44
AVPR1A P37288 2/20 0.43
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7334113 0.94 AVPR2 (0.54) AVPR2ROCK2TP53SHMT2AVPR1A
SCHEMBL7342906 0.94 AVPR2 (0.49) AVPR2ROCK2TP53SHMT2AVPR1A
SCHEMBL7344625 0.91 AVPR2 (0.49) AVPR2TP53SHMT2AVPR1ALMNA
SCHEMBL7343152 0.91 AVPR2 (0.54) AVPR2TP53AVPR1A
SCHEMBL7343689 0.91 AVPR2 (0.48) AVPR2TP53SHMT2AVPR1ALMNA
SCHEMBL7339437 0.87 TP53 (0.44) AVPR2TP53SHMT2AVPR1ALMNA
SCHEMBL7334015 0.86 AVPR2 (0.44) AVPR2TP53SHMT2AVPR1ALMNA
SCHEMBL7342384 0.85 AVPR2 (0.61) AVPR2AVPR1A
SCHEMBL7339456 0.84 AVPR2 (0.56) AVPR2TP53AVPR1A
SCHEMBL7343088 0.83 AVPR2 (0.48) AVPR2TP53SHMT2AVPR1ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed