SCHEMBL7400845

SCHEMBL7400845

O=C(CCn1cnc2c(=O)[nH]cnc21)NCc1ccc2c(c1)OCO2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.54
HPGD P15428 2/20 0.54
POLB P06746 1/20 0.54
ALDH1A1 P00352 3/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
HTT P42858 1/20 0.48
TP53 P04637 2/20 0.48
LMNA P02545 1/20 0.48
TSHR P16473 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MAPK1 P28482 2/20 0.48
USP2 O75604 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7568100 0.86 TDP1 (0.56) TDP1HPGDPOLBALDH1A1L3MBTL1
SCHEMBL7398812 0.75 HPRT1 (0.48) TDP1HPGDPOLBL3MBTL1MEN1
SCHEMBL7399609 0.74 HPRT1 (0.56)
SCHEMBL7376553 0.74 HPRT1 (0.47) HPGDALDH1A1LMNAMEN1KMT2A
SCHEMBL7399531 0.73 HPRT1 (0.55)
SCHEMBL7398541 0.73 HPRT1 (0.55)
SCHEMBL179082 0.73 HPGD (0.73) TDP1HPGDPOLBALDH1A1L3MBTL1
SCHEMBL7397072 0.73 HPRT1 (0.59)
SCHEMBL7392166 0.73 HPRT1 (0.54)
SCHEMBL7222745 0.72 HPGD (0.69) TDP1HPGDPOLBALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0522082-B1 MULTI-FUNCTIONAL PHARMACEUTICAL COMPOUNDS AND METHODS OF USE GLASKY ALVIN J (US) 1997-07-02 EP disclosed
EP-0522082-A4 MULTI-FUNCTIONAL PHARMACEUTICAL COMPOUNDS AND METHODS OF USE 1993-06-09 EP disclosed
EP-0522082-A1 MULTI-FUNCTIONAL PHARMACEUTICAL COMPOUNDS AND METHODS OF USE. GLASKY ALVIN J (US) 1993-01-13 EP disclosed
US-5091432-A Synergistic SPECTRUM PHARMACEUTICALS, INC. 1992-02-25 US disclosed
WO-1991014434-A1 MULTI-FUNCTIONAL PHARMACEUTICAL COMPOUNDS AND METHODS OF USE GLASKY ALVIN J (US) 1991-10-03 WO disclosed