SCHEMBL7401632

SCHEMBL7401632

C=C(CC(=O)Nc1ccc(C#N)cc1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SAE1 Q9UBE0 1/20 0.51
UBA2 Q9UBT2 1/20 0.51
MAPT P10636 5/20 0.49
LMNA P02545 2/20 0.49
TSHR P16473 1/20 0.49
HTT P42858 1/20 0.49
NLRP3 Q96P20 1/20 0.49
KMT2A Q03164 4/20 0.47
POLB P06746 4/20 0.47
MEN1 O00255 3/20 0.47
KDM4E B2RXH2 1/20 0.47
PKM P14618 1/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 1/20 0.47
IL18 Q14116 1/20 0.47
PAX8 Q06710 1/20 0.47
GAA P10253 2/20 0.47
ALDH1A1 P00352 3/20 0.45
FNTA P49354 1/20 0.45
FNTB P49356 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20941638 0.84 SAE1 (0.62) SAE1UBA2MAPTLMNATSHR
SCHEMBL841012 0.83 SAE1 (0.57) SAE1UBA2MAPTLMNATSHR
SCHEMBL5175525 0.80 CYP1A1 (0.58) MAPTTSHRKMT2APOLBMEN1
SCHEMBL4337854 0.79 EPHX2 (0.55) MAPTTSHRHTTKMT2AMEN1
SCHEMBL4900622 0.78 KMT2A (0.58) MAPTLMNATSHRHTTKMT2A
SCHEMBL4905462 0.78 POLB (0.69) MAPTHTTKMT2APOLBMEN1
SCHEMBL11260465 0.78 MAPT (0.57) SAE1UBA2MAPTLMNATSHR
SCHEMBL8044037 0.78 SAE1 (0.59) SAE1UBA2MAPTLMNATSHR
SCHEMBL20941635 0.77 MAPT (0.75) SAE1UBA2MAPTLMNATSHR
SCHEMBL20941549 0.77 SAE1 (0.54) SAE1UBA2MAPTLMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939418-A ANTICOAGULANT THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1999-08-17 US disclosed
EP-0874629-A4 ISOXAZOLINE, ISOTHIAZOLINE AND PYRAZOLINE FACTOR Xa INHIBITORS DU PONT MERCK PHARMA (US) 1999-08-04 EP disclosed
EP-0874629-A1 ISOXAZOLINE, ISOTHIAZOLINE AND PYRAZOLINE FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-11-04 EP disclosed
WO-1997023212-A1 ISOXAZOLINE, ISOTHIAZOLINE AND PYRAZOLINE FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-07-03 WO disclosed