SCHEMBL740176

SCHEMBL740176

COc1cc2c(c(-c3ccc(C(F)(F)F)cc3)c1OC)CN(CCCCC(C)C(=O)O)C2=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.41
AKR1C2 P52895 4/20 0.41
PPARD Q03181 4/20 0.36
PPARA Q07869 4/20 0.36
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
BACE1 P56817 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL450867 0.87 KDM4E (0.42) AKR1C3AKR1C2PPARDPPARAKDM4E
SCHEMBL452313 0.84 S1PR1 (0.36) AKR1C3AKR1C2KDM4ENPC1TP53
SCHEMBL437104 0.75 KDM4E (0.47) KDM4EMAPTTSHRSMN1; SMN2ALDH1A1
SCHEMBL447230 0.69 HDAC1 (0.54)
SCHEMBL450113 0.69 HDAC1 (0.36) KDM4EALDH1A1HPGD
SCHEMBL25904813 0.65 CNR2 (0.47) PPARDPPARA
SCHEMBL25323579 0.64 CNR2 (0.46)
SCHEMBL25326358 0.63 CNR2 (0.47) PPARDPPARA
SCHEMBL24306488 0.62 CNR2 (0.42) HSD17B10ALDH1A1
SCHEMBL25325057 0.61 CNR2 (0.45) PPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429987-A2 AMIDE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING SAME Korea Research Institute Of Chemical Technology (KR) 2012-03-21 EP disclosed