SCHEMBL7404668

SCHEMBL7404668

COC(=O)N[C@H](C(=O)NC(Cc1ccccc1)C(O)CN(N)Cc1ccc(-c2ccccn2)cc1)C(C)C

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT1A1 P22309 3/20 0.66
MLNR O43193 1/20 0.66
NR1I2 O75469 1/20 0.66
SLCO2B1 O94956 1/20 0.66
ABCB11 O95342 1/20 0.66
ABCB1 P08183 1/20 0.66
CCKAR P32238 1/20 0.66
OPRK1 P41145 1/20 0.66
GHSR Q92847 1/20 0.66
SLCO1B3 Q9NPD5 1/20 0.66
ABCG2 Q9UNQ0 1/20 0.66
SLCO1B1 Q9Y6L6 1/20 0.66
KCNH2 Q12809 1/20 0.53
CA2 P00918 2/20 0.47
CTSD P07339 4/20 0.47
CYP3A4 P08684 1/20 0.47
PSEN1 P49768 3/20 0.45
PSEN2 P49810 3/20 0.45
APH1B Q8WW43 3/20 0.45
NCSTN Q92542 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7404665 1.00 UGT1A1 (0.66) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL6041 0.99 UGT1A1 (0.65) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL6157360 0.99 UGT1A1 (0.65) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL8091155 0.94 UGT1A1 (0.61) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL8091153 0.94 UGT1A1 (0.61) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL5829 0.93 UGT1A1 (0.60) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL6201 0.93 UGT1A1 (0.60) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL6156161 0.93 UGT1A1 (0.60) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL5793 0.90 UGT1A1 (0.55) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL6157073 0.90 UGT1A1 (0.55) UGT1A1MLNRNR1I2SLCO2B1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900210-A1 ANTIVIRALLY ACTIVE HETEROCYCLIC AZAHEXANE DERIVATIVES Novartis AG (CH) 1999-03-10 EP disclosed
WO-1997040029-A1 ANTIVIRALLY ACTIVE HETEROCYCLIC AZAHEXANE DERIVATIVES NOVARTIS AG (CH) 1997-10-30 WO disclosed