SCHEMBL7405774

SCHEMBL7405774

Cc1cn(-c2cc(F)cc(N)c2N)cn1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 1/20 0.42
PSEN1 P49768 14/20 0.37
PSEN2 P49810 13/20 0.37
APH1B Q8WW43 13/20 0.37
NCSTN Q92542 13/20 0.37
APH1A Q96BI3 13/20 0.37
PSENEN Q9NZ42 13/20 0.37
SCD O00767 1/20 0.35
KCNH2 Q12809 1/20 0.34
CYP2E1 P05181 1/20 0.34
CYP2A6 P11509 1/20 0.34
APP P05067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL970409 0.81 PSEN1 (0.43) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL12247676 0.77 PSEN1 (0.38) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL12886318 0.73 CYP2E1 (0.42) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL12247672 0.73 PSEN1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1616928 0.71 NR2E1 (0.46) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL7402126 0.70 IDO1 (0.49)
SCHEMBL27819262 0.69 GAA (0.48) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL909015 0.69 PSEN1 (0.43) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL2790568 0.69 NR2E1 (0.57) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL30661672 0.68 NR2E1 (0.37) NR2E1PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999026932-A1 BY AMIDINO GROUP SUBSTITUTED HETEROCYCLIC DERIVATIVES AND THEIR USE AS ANTICOAGULANTS AXYS PHARMACEUTICALS, INC. (US) 1999-06-03 WO disclosed