SCHEMBL740784

SCHEMBL740784

COCCCc1cccc(N)c1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.38
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP2C9 P11712 1/20 0.34
ALOX5 P09917 1/20 0.33
PTGS2 P35354 1/20 0.33
ALDH1A1 P00352 3/20 0.32
ADRA2B P18089 1/20 0.32
PTGS1 P23219 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TSHR P16473 2/20 0.32
CYP3A4 P08684 1/20 0.32
PIK3CA P42336 1/20 0.32
TYMS P04818 1/20 0.32
KDM4E B2RXH2 2/20 0.32
TLR7 Q9NYK1 1/20 0.32
HPGD P15428 1/20 0.32
RCE1 Q9Y256 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28220304 0.89 CD44 (0.40) CD44CYP1A2CYP2C19CYP2C9ALDH1A1
SCHEMBL3078026 0.85 CYP1A2 (0.40) CYP1A2CYP2C19CYP2C9ALDH1A1ADRA2B
SCHEMBL15771668 0.82 TAAR1 (0.38) ADRA2BHPGDTAAR1DGAT2
SCHEMBL3065473 0.79 CYP1A2 (0.39) CYP1A2CYP2C19CYP2C9ALOX5PTGS2
SCHEMBL659538 0.79 TLR8 (0.42) CD44CYP1A2CYP2C19CYP2C9ALOX5
SCHEMBL15771442 0.77 TAAR1 (0.37) ALOX5PTGS2ADRA2BTDP1HPGD
SCHEMBL3482721 0.77 CD44 (0.46) CD44ALDH1A1TDP1TSHRCYP3A4
SCHEMBL4763408 0.77 BID (0.47) ALOX5PTGS2KDM4E
SCHEMBL4038330 0.76 CD44 (0.43) CD44ALDH1A1ADRA2BPTGS1TDP1
SCHEMBL30645137 0.76 CD44 (0.43) CD44ALDH1A1ADRA2BPTGS1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-7868036-B2 Organic compounds NOVARTIS AG (CH) 2011-01-11 US disclosed
EP-1725530-A1 ORGANIC COMPOUNDS Speedel Experimenta AG (CH) 2006-11-29 EP disclosed
WO-2005090304-A1 ORGANIC COMPOUNDS SPEEDEL EXPERIMENTA AG (CH) 2005-09-29 WO disclosed