SCHEMBL740852

SCHEMBL740852

NC(=O)CCn1c(C2CCCN(C(=O)CC(N)Cc3ccc(-c4ccccc4)cc3)C2)nc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.49
POLB P06746 1/20 0.49
HRH1 P35367 9/20 0.47
CYP2D6 P10635 7/20 0.47
KCNH2 Q12809 9/20 0.43
CHRM1 P11229 3/20 0.43
HTR2B P41595 1/20 0.42
GRM2 Q14416 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740851 1.00 USP2 (0.49) USP2POLBHRH1CYP2D6KCNH2
SCHEMBL742622 0.94 HRH1 (0.47) USP2POLBHRH1CYP2D6KCNH2
SCHEMBL739835 0.94 HRH1 (0.47) USP2POLBHRH1CYP2D6KCNH2
SCHEMBL739836 0.94 HRH1 (0.47) USP2POLBHRH1CYP2D6KCNH2
SCHEMBL742623 0.94 HRH1 (0.47) USP2POLBHRH1CYP2D6KCNH2
SCHEMBL739730 0.92 KCNH2 (0.52) USP2POLBHRH1CYP2D6KCNH2
SCHEMBL739731 0.92 KCNH2 (0.52) USP2POLBHRH1CYP2D6KCNH2
SCHEMBL738684 0.92 HRH1 (0.44) USP2POLBHRH1CYP2D6KCNH2
SCHEMBL738685 0.92 HRH1 (0.44) USP2POLBHRH1CYP2D6KCNH2
SCHEMBL741488 0.92 HRH1 (0.43) USP2POLBHRH1CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed