SCHEMBL7408574

SCHEMBL7408574

Cc1cc(C(=O)Nc2ccc(-n3nnnc3C(F)(F)F)cc2)n(-c2cccc(CN)c2)n1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 9/20 0.59
F10 P00742 8/20 0.57
F2 P00734 7/20 0.57
PRSS1 P07477 7/20 0.57
PRSS2 P07478 7/20 0.57
PRSS3 P35030 7/20 0.57
TSHR P16473 1/20 0.50
CARM1 Q86X55 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19710439 0.79 TSHR (0.74) KLKB1F10F2PRSS1PRSS2
SCHEMBL3831539 0.78 F10 (0.58) KLKB1F10F2PRSS1PRSS2
SCHEMBL3832891 0.78 KLKB1 (0.72) KLKB1F10F2PRSS1PRSS2
SCHEMBL18622996 0.76 KLKB1 (0.65) KLKB1F10F2PRSS1PRSS2
SCHEMBL7395467 0.76 F10 (0.60) KLKB1F10F2PRSS1PRSS2
SCHEMBL18623001 0.75 KLKB1 (0.66) KLKB1F10F2PRSS1PRSS2
SCHEMBL18623002 0.75 KLKB1 (0.66) KLKB1F10F2PRSS1PRSS2
SCHEMBL3833307 0.75 F10 (0.56) KLKB1F10F2PRSS1PRSS2
SCHEMBL18623006 0.73 KLKB1 (0.64) KLKB1F10F2PRSS1PRSS2
SCHEMBL18623107 0.73 KLKB1 (0.60) KLKB1F10F2PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946508-A1 NITROGEN CONTAINING HETEROAROMATICS AS FACTOR Xa INHIBITORS Du Pont Pharmaceuticals Company (US) 1999-10-06 EP disclosed
WO-1998028269-A1 NITROGEN CONTAINING HETEROAROMATICS AS FACTOR Xa INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 1998-07-02 WO disclosed