SCHEMBL740945

SCHEMBL740945

CC(C)(C)OC(=O)N1CCCC(C(=O)Nc2c(N)cccc2Cl)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 3/20 0.48
ABL1 P00519 1/20 0.48
RIN1 Q13671 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
USP30 Q70CQ3 2/20 0.46
PTPN2 P17706 1/20 0.46
PTPN1 P18031 1/20 0.46
PTPN6 P29350 1/20 0.46
HSD11B1 P28845 1/20 0.45
RHOA P61586 2/20 0.43
PARP1 P09874 2/20 0.43
PARP2 Q9UGN5 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
ACKR3 P25106 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740946 1.00 STS (0.48) STSABL1RIN1MEN1KMT2A
SCHEMBL742851 0.86 STS (0.48) STSABL1RIN1MEN1KMT2A
SCHEMBL742852 0.86 STS (0.48) STSABL1RIN1MEN1KMT2A
SCHEMBL17533942 0.84 HDAC1 (0.62) ABL1RIN1MEN1KMT2AALDH1A1
SCHEMBL762580 0.84 HDAC1 (0.62) ABL1RIN1MEN1KMT2AALDH1A1
SCHEMBL19378084 0.84 HDAC1 (0.62) ABL1RIN1MEN1KMT2AALDH1A1
SCHEMBL740750 0.84 RHOA (0.47) KMT2AALDH1A1RHOARAB9AHDAC1
SCHEMBL16895918 0.82 USP30 (0.49) STSABL1RIN1MEN1KMT2A
SCHEMBL16791247 0.82 USP30 (0.49) STSABL1RIN1MEN1KMT2A
SCHEMBL2636168 0.81 STS (0.52) STSALDH1A1MAPTUSP30PTPN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed