SCHEMBL741107

SCHEMBL741107

OC1(F)CCC(Oc2ccc(-c3ccn4c(CC5CC5)nnc4c3C(F)(F)F)cc2Cl)CC1

nearest known ligand 0.80

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 20/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10323148 0.89 GRM2 (1.00) GRM2
SCHEMBL10325106 0.89 GRM2 (1.00) GRM2
SCHEMBL10323147 0.89 GRM2 (1.00) GRM2
SCHEMBL741461 0.87 GRM2 (1.00) GRM2
SCHEMBL743143 0.78 GRM2 (1.00) GRM2
SCHEMBL10325109 0.77 GRM2 (1.00) GRM2
SCHEMBL10325107 0.77 GRM2 (1.00) GRM2
SCHEMBL10325108 0.77 GRM2 (1.00) GRM2
SCHEMBL30795377 0.77 GRM2 (1.00) GRM2
SCHEMBL742376 0.77 GRM2 (1.00) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430021-A1 7-ARYL-1,2,4-TRIAZOLOÝ4,3-A¨PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS Janssen Pharmaceuticals Inc. (US) 2012-03-21 EP disclosed
WO-2010130423-A1 7-ARYL-1,2,4-TRIAZOLO[4,3-A]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS ORTHO-MCNEIL-JANSSEN PHARMACEUTICALS, INC (US) 2010-11-18 WO disclosed