SCHEMBL7413757

SCHEMBL7413757

NC(Cc1ccc2nc(-c3c(Cl)cccc3Cl)oc2c1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.57
ITGA4 P13612 3/20 0.57
ITGB7 P26010 3/20 0.57
PKM P14618 2/20 0.48
PTPRA P18433 1/20 0.44
PTPRB P23467 1/20 0.44
SLC7A5 Q01650 3/20 0.43
HIF1A Q16665 2/20 0.42
PTGS1 P23219 2/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
EGFR P00533 1/20 0.42
LCK P06239 1/20 0.42
FYN P06241 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ALOX15 P16050 1/20 0.42
HTR2A P28223 1/20 0.42
PTGS2 P35354 1/20 0.42
RECQL P46063 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413758 1.00 ITGB1 (0.57) ITGB1ITGA4ITGB7PKMPTPRA
SCHEMBL7420912 0.91 ITGB1 (0.68) ITGB1ITGA4ITGB7PKMPTPRA
SCHEMBL7420913 0.91 ITGB1 (0.68) ITGB1ITGA4ITGB7PKMPTPRA
SCHEMBL5130333 0.81 ITGB1 (0.85) ITGB1ITGA4ITGB7ITGAV
SCHEMBL5125672 0.78 ITGB1 (0.86) ITGB1ITGA4ITGB7ITGAV
SCHEMBL3314275 0.77 ITGB1 (0.67) ITGB1PKMSLC7A5HIF1APTGS1
SCHEMBL3318103 0.77 ITGB1 (0.67) ITGB1PKMSLC7A5HIF1APTGS1
SCHEMBL5127850 0.76 ITGB1 (0.44) ITGB1ITGA4ITGB7KDM4EALOX15
SCHEMBL460247 0.75 TTR (0.69) ITGB1ITGA4ITGB7TTRALB
SCHEMBL23729861 0.74 TTR (0.54) PKMSLC7A5TTRALBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420418-B1 INHIBITION AND PREVENTION OF LEUKOCYTE ADHESION; USED TO TREAT ADHESION-MEDIATED DISEASES SUCH AS ASTHMA, ALLERGIC RHINITIS, MULTIPLE SCLEROSIS; ATHEROSCLEROSIS, AND INFLAMMATORY BOWEL DISEASE MERCK & CO., INC. 2002-07-16 US disclosed
WO-2001012183-A1 HETEROCYCLE AMIDES AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 2001-02-22 WO disclosed