SCHEMBL7414764

SCHEMBL7414764

CN1Cc2nc(Br)cnc2N(C)C1=O

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.33
BIRC2 Q13490 1/20 0.33
CASP3 P42574 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414097 0.72 XIAP (0.50) XIAPBIRC2
SCHEMBL7416621 0.71 XIAP (0.40) XIAPBIRC2
SCHEMBL7421949 0.71 BRD4 (0.40) CASP3
SCHEMBL19508034 0.66 FGFR4 (0.40)
SCHEMBL15595097 0.64 MTOR (0.34)
SCHEMBL6619181 0.62 FGFR4 (0.37)
SCHEMBL18824526 0.60 MEN1 (0.45)
SCHEMBL7415042 0.59 BRD4 (0.51) XIAPBIRC2
SCHEMBL13826643 0.59 XIAP (0.50) XIAPBIRC2
SCHEMBL21932324 0.58 XIAP (0.38) XIAPBIRC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5002944-A Compounds having cardiotonic activity RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-03-26 US disclosed
EP-0333727-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (a Delaware corporation) (US) 1989-09-27 EP disclosed
US-4859672-A Pyrido[2,3-d]pyrimidinone and imidazo[4,5-b]pyrimidinone RORER PHARMACEUTICAL CORPORATION (US) 1989-08-22 US disclosed
WO-1988003025-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (US) 1988-05-05 WO disclosed