SCHEMBL7415487

SCHEMBL7415487

O=C1Nc2ccc(Cl)cc2Cc2sccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.55
CES1 P23141 2/20 0.45
TGM2 P21980 2/20 0.45
CMA1 P23946 1/20 0.44
CHEK1 O14757 1/20 0.43
PPOX P50336 1/20 0.41
PGR P06401 1/20 0.40
TDP2 O95551 2/20 0.39
CCNB2 O95067 1/20 0.39
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
GSK3B P49841 1/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
LRRK2 Q5S007 4/20 0.38
HTR5A P47898 3/20 0.38
ADRA2A P08913 2/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7406111 0.90 AHR (0.57) AHRCES1TGM2CMA1CHEK1
SCHEMBL7411028 0.80 AHR (0.52) AHRCES1TDP2GSK3BLRRK2
SCHEMBL154614 0.72 AHR (1.00) AHRCMA1PGRTDP2HTR5A
SCHEMBL14809527 0.71 AHR (0.70) AHRCES1TGM2CMA1CHEK1
SCHEMBL8584695 0.70 AHR (0.86) AHRCMA1PGRTDP2CCNB2
SCHEMBL11105121 0.70 CHEK1 (0.53) AHRCES1TGM2CMA1CHEK1
SCHEMBL31139641 0.69 CES1 (0.77) CES1TGM2CHEK1PPOXLRRK2
SCHEMBL7016454 0.69 AHR (0.61) AHRCES1TGM2CMA1CHEK1
SCHEMBL11536683 0.68 CHEK1 (0.61) AHRCES1TGM2CMA1CHEK1
SCHEMBL11538675 0.67 AHR (0.59) AHRCMA1CHEK1PGRHTR5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3962248-A PROCESS FOR MAKING 11-PIPERAZINO-DIAZEPINES, OXAZEPINES, THIAZEPINES AND AZEPINES SANDOZ, INC. (US) 1976-06-08 US disclosed