SCHEMBL7416359

SCHEMBL7416359

CC(C)(C)OC(=O)N1CC[C@@H]1COS(=O)(=O)Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
STS P08842 1/20 0.53
NR1H2 P55055 2/20 0.48
NR1H3 Q13133 2/20 0.48
NPSR1 Q6W5P4 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KLK7 P49862 1/20 0.43
HCRTR2 O43614 1/20 0.42
PKM P14618 2/20 0.41
GPR119 Q8TDV5 2/20 0.41
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7670460 1.00 STS (0.53) STSNR1H2NR1H3NPSR1ALDH1A1
SCHEMBL7414543 1.00 STS (0.53) STSNR1H2NR1H3NPSR1ALDH1A1
SCHEMBL29407129 0.93 STS (0.51) STSNR1H2NR1H3NPSR1ALDH1A1
SCHEMBL30365707 0.92 STS (0.48) STSNR1H2NR1H3NPSR1ALDH1A1
SCHEMBL6870558 0.83 NPSR1 (0.47) STSNPSR1ALDH1A1MAPTKLK7
SCHEMBL1879011 0.83 STS (0.63) STSPKMGPR119GAAJAK2
SCHEMBL7414412 0.83 STS (0.47) STSNR1H2NR1H3KLK7HCRTR2
SCHEMBL7921498 0.82 KLK7 (0.47) STSNR1H2NR1H3KLK7PKM
SCHEMBL7921496 0.82 KLK7 (0.47) STSNR1H2NR1H3KLK7PKM
SCHEMBL7667825 0.81 NR1H2 (0.41) STSNR1H2NR1H3NPSR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950057-B1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS ABBOTT LAB (US) 2002-11-13 EP disclosed
US-6403575-B1 ANTI-INFLAMMATORIES ABBOTT LABORATORIES 2002-06-11 US disclosed
EP-1047690-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-11-02 EP disclosed
US-6133253-A NEURONAL CELL DEATH PREVENTORS AND ANTI-INFLAMMATORIES ABBOTT LABORATORIES (US) 2000-10-17 US disclosed
EP-0950057-A1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS Abbott Laboratories (US) 1999-10-20 EP disclosed
WO-1999032480-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1999-07-01 WO disclosed
WO-1998025920-A1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS ABBOTT LABORATORIES (US) 1998-06-18 WO disclosed