SCHEMBL7416729

SCHEMBL7416729

CSc1sc(C(=O)N(C)C)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.64
LMNA P02545 1/20 0.64
GABRG2 P18507 10/20 0.52
GABRB3 P28472 10/20 0.52
GABRA5 P31644 10/20 0.52
GABRA3 P34903 9/20 0.52
GABRA1 P14867 8/20 0.52
GABRA2 P47869 8/20 0.52
LRRK2 Q5S007 2/20 0.46
CCNC P24863 1/20 0.46
CDK8 P49336 1/20 0.46
CDK19 Q9BWU1 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7452104 0.85 NPSR1 (0.68) NPSR1LMNAGABRG2GABRB3GABRA5
SCHEMBL4401833 0.85 NPSR1 (0.68) NPSR1LMNAGABRG2GABRB3GABRA5
SCHEMBL7415050 0.84 NPSR1 (0.56) NPSR1LMNAGABRG2GABRB3GABRA5
SCHEMBL7459195 0.81 NPSR1 (0.75) NPSR1LMNAGABRG2GABRB3GABRA5
SCHEMBL7458560 0.81 NPSR1 (0.64) NPSR1LMNAGABRG2GABRB3GABRA5
SCHEMBL4931496 0.80 NPSR1 (0.62) NPSR1LMNAGABRG2GABRB3GABRA5
SCHEMBL7459881 0.79 NPSR1 (0.61) NPSR1LMNAGABRG2GABRB3GABRA5
SCHEMBL7459875 0.79 NPSR1 (0.61) NPSR1LMNAGABRG2GABRB3GABRA5
SCHEMBL7463997 0.79 NPSR1 (0.61) NPSR1LMNAGABRG2GABRB3GABRA5
SCHEMBL7416513 0.78 NPSR1 (0.60) NPSR1LMNAGABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156787-A Substituted thienlycyclohexanone derivatives for enhancing cognition MERCK SHARP & DOHME LIMITED (GB) 2000-12-05 US disclosed
US-6143773-A Substituted thienobenzisoxazole derivatives for enhancing cognition MERCK SHARP & DOHME LIMITED (GB) 2000-11-07 US disclosed
WO-1995007885-A1 DERIVATIVES OF 2-AMINO-1,2,3,4-TETRAHYDRONAPHTHALENE ACTIVE ON THE CARDIOVASCULAR SYSTEM ZAMBON GROUP S.P.A. (IT) 1995-03-23 WO disclosed